2hz4 A 2.8 BS01 4ST A 1 W261 Y264 L266 K294 L302 W23 Y26 L28 K56 L64 D363 A365 R367 N368 D381 P402 D125 A127 R129 N130 D143 P164 2.7.10.2 0004672,0004713,0005524,0006468 -logKd/Ki=5.47, IC50=3425nM P00519 17164530 501 KWEMERTDITMKHKLGEVYEGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQES 2hz4 A 2.8 BS02 4ST C 1 Y342 F497 Q498 S500 Y104 F259 Q260 S262 D363 A365 R367 N368 D381 P402 D125 A127 R129 N130 D143 P164 2.7.10.2 0004672,0004713,0005524,0006468 -logKd/Ki=5.47, IC50=3425nM P00519 17164530 501 KWEMERTDITMKHKLGEVYEGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQES 2hz4 C 2.8 BS01 4ST A 1 F497 Q498 S500 F256 Q257 S259 D363 A365 R367 N368 D381 P402 D122 A124 R126 N127 D140 P161 2.7.10.2 0004672,0004713,0005524,0006468 P00519 17164530 501 KWEMERTDITMKHKLGEVYEGVWKKYTVAVKTLKDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQES