2hyy A 2.4 BS01 STI A 1 L248 Y253 A269 K271 E286 V289 M290 T315 F317 M318 I360 H361 L370 A380 D381 F382 L14 Y19 A35 K37 E51 V54 M55 T80 F82 M83 I125 H126 L135 A145 D146 F147 D363 A365 R367 N368 D381 P402 D128 A130 R132 N133 D146 P167 2.7.10.2 0004672,0004713,0005524,0006468 ic50=170nM -logKd/Ki=6.77, IC50=170nM IC50=38nM, Kd=44nM, Ki=13nM, EC50=7e+1nM P00519 17164530 600 WEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQ