2gqg A 2.4 BS01 1N1 A 1 L248 A269 K271 E286 M290 V299 I313 T315 F317 M318 T319 Y320 G321 L370 L26 A47 K49 E64 M68 V77 I91 T93 F95 M96 T97 Y98 G99 L148 D363 A365 R367 N368 D381 P402 D141 A143 R145 N146 D159 P180 2.7.10.2 0004672,0004713,0005524,0006468 IC50=3.1nM, Kd=1.2nM, EC50=0.040000nM P00519 16740718 501 GAMDPSSPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQES