2gg3 A 1.45 BS01 CO A 1 D108 H171 T202 E204 E235 D107 H170 T201 E203 E234 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H78 D96 D107 H170 R174 H177 Q181 E203 N207 Q232 E234 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0046914,0070006 P0AE18 17120228 301 AISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHDE 2gg3 A 1.45 BS02 CO A 2 D97 D108 E235 D96 D107 E234 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H78 D96 D107 H170 R174 H177 Q181 E203 N207 Q232 E234 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0046914,0070006 P0AE18 17120228 302 AISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHDE 2gg3 A 1.45 BS03 U13 A 1 Y62 H63 H79 D97 D108 H171 F177 H178 E204 W221 E235 Y61 H62 H78 D96 D107 H170 F176 H177 E203 W220 E234 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H78 D96 D107 H170 R174 H177 Q181 E203 N207 Q232 E234 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0046914,0070006 ic50=0.58uM -logKd/Ki=6.24, IC50=0.58uM IC50=580nM P0AE18 17120228 501 AISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHDE