2fgi A 2.5 BS01 PD1 A 1 L484 G485 V492 A512 K514 M535 I545 V561 Y563 A564 S565 G567 L630 A640 D641 L21 G22 V24 A40 K42 M63 I73 V89 Y91 A92 S93 G95 L144 A154 D155 D623 A625 R627 N628 D641 D137 A139 R141 N142 D155 2.7.10.1 0004672,0004713,0005007,0005524,0006468 Ki=36.4nM -logKd/Ki=7.34, Ki=45.2nM IC50=22nM, EC50=21nM P11362 9774334 1001 ELPEDPRWELPRDRLVLGKPLGQVVLAEAIGLPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRPPQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLADIHHIDYYKKTNGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALTS