2e9u A 2.0 BS01 A25 A 1 L15 A36 V68 L84 E85 Y86 C87 G90 L137 S147 L14 A35 V67 L83 E84 Y85 C86 G89 L136 S146 D130 K132 E134 N135 D148 T170 D129 K131 E133 N134 D147 T169 2.7.11.1 0000077,0004672,0004674,0005524,0006468 -logKd/Ki=8.10, Ki=7.94nM IC50=10nM O14757 1001 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRAVDCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK