2d0t A 2.3 BS01 HEM A 1 F163 V170 F214 I217 F226 S263 A264 F270 R343 H346 I349 Y353 I354 L384 V391 F152 V159 F203 I206 F215 S252 A253 F259 R332 H335 I338 Y342 I343 L354 V361 1.13.11.52 0002376,0002666,0002678,0002830,0004833,0005737,0005829,0006569,0006954,0007565,0009055,0016702,0019441,0019805,0020037,0030485,0032421,0032496,0032693,0032735,0033555,0033754,0034276,0034354,0036269,0042098,0042130,0043065,0046006,0046872,0051213,0070233,0070234 P14902 16477023 404 SKEYHIDEEVGFALPNPQENLPDFYNDWMFIAKHLPDLIESGQLRERVEKLNMLSIDHLTDHKSQRLARLVLGCITMAYVWGKGHGDVRKVLPRNIAVPYCQLSKKLELPPILVYADCVLANWKKKDPNKPLTYENMDVLFSFRDGDCSKGFFLVSLLVEIAAASAIKVIPTVFKAMQMQERDTLLKALLEIASCLEKALQVFHQIHDHVNPKAFFSVLRIYLSGWKGNPQLSDGLVYEGFWEDPKEFAGGSAGQSSVFQCFDVLLGIQQTAGGGHAAQFLQDMRRYMPPAHRNFLCSLESNPSVREFVLSKGDAGLREAYDACVKALVSLRSYHLQIVTKYILIPASQGGTDLMNFLKTVRSTTEKSLLKEG 2d0t A 2.3 BS02 PIM A 1 V130 F163 F164 S167 S263 A264 V119 F152 F153 S156 S252 A253 1.13.11.52 0002376,0002666,0002678,0002830,0004833,0005737,0005829,0006569,0006954,0007565,0009055,0016702,0019441,0019805,0020037,0030485,0032421,0032496,0032693,0032735,0033555,0033754,0034276,0034354,0036269,0042098,0042130,0043065,0046006,0046872,0051213,0070233,0070234 IC50=48000nM P14902 16477023 501 SKEYHIDEEVGFALPNPQENLPDFYNDWMFIAKHLPDLIESGQLRERVEKLNMLSIDHLTDHKSQRLARLVLGCITMAYVWGKGHGDVRKVLPRNIAVPYCQLSKKLELPPILVYADCVLANWKKKDPNKPLTYENMDVLFSFRDGDCSKGFFLVSLLVEIAAASAIKVIPTVFKAMQMQERDTLLKALLEIASCLEKALQVFHQIHDHVNPKAFFSVLRIYLSGWKGNPQLSDGLVYEGFWEDPKEFAGGSAGQSSVFQCFDVLLGIQQTAGGGHAAQFLQDMRRYMPPAHRNFLCSLESNPSVREFVLSKGDAGLREAYDACVKALVSLRSYHLQIVTKYILIPASQGGTDLMNFLKTVRSTTEKSLLKEG