2cni A 2.0 BS01 IZF A 1 Y20 R24 Y46 D48 D181 F182 C215 S216 A217 I219 G220 R221 R254 M258 G259 Q262 L299 Y20 R24 Y46 D48 D181 F182 C215 S216 A217 I219 G220 R221 R254 M258 G259 Q262 L299 D181 C215 R221 S222 Q262 D181 C215 R221 S222 Q262 3.1.3.48 0004725,0006470,0016311 ic50=21nM -logKd/Ki=7.68, IC50=21nM P18031 17028182 1301 MEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHEDL