2cmc A 2.2 BS01 DFM A 1 Y46 R47 D48 V49 F182 C215 S216 A217 I219 G220 R221 Q262 K279 F280 Y51 R52 D53 V54 F187 C220 S221 A222 I224 G225 R226 Q267 K284 F285 D181 C215 R221 S222 Q262 D186 C220 R226 S227 Q267 3.1.3.48 0004725,0006470,0016311 ic50=1750nM -logKd/Ki=5.76, IC50=1.75uM IC50=1750nM P18031 16916797 1281 HHHHHHEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKF