2bge A 1.8 BS01 T2D A 1 Y46 S151 D181 F182 C215 S216 A217 I219 G220 R221 Q262 E297 Y46 S151 D181 F182 C215 S216 A217 I219 G220 R221 Q262 E297 D181 C215 R221 S222 Q262 D181 C215 R221 S222 Q262 3.1.3.48 0004725,0006470,0016311 ic50=1608uM -logKd/Ki=2.80, IC50=1.6mM IC50=1600000nM P18031 15863305 1298 MEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHE