2bgd A 2.4 BS01 T1D A 1 Y46 V49 K150 F182 C215 S216 A217 I219 G220 R221 E297 Y46 V49 K147 F179 C212 S213 A214 I216 G217 R218 E294 D181 C215 R221 S222 Q262 D178 C212 R218 S219 Q259 3.1.3.48 0004725,0006470,0016311 ic50=2.47uM -logKd/Ki=5.00, Kd<10uM IC50=2500nM P18031 15863305 1298 MEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHE