2ayr A 1.9 BS01 L4G A 1 M343 L346 T347 A350 D351 E353 W383 L387 R394 M421 I424 H524 L525 K529 M38 L41 T42 A45 D46 E48 W78 L82 R89 M116 I119 H219 L220 K224 ? Ki=0.51nM -logKd/Ki=9.29, Ki=0.51nM Ki=0.47nM, EC50=10.7nM P03372 16250633 201 LALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLESAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKSVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLSSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKSKNVVPLYDLLLEMLDAHRLHA