1zrz A 3.0 BS01 BI1 A 1 I251 G252 V259 A272 K274 E324 Y325 V326 D373 L376 T386 D387 I12 G13 V20 A33 K35 E85 Y86 V87 D134 L137 T147 D148 D369 K371 N374 D387 T407 D130 K132 N135 D148 T168 2.7.11.13 0004672,0004674,0004697,0005524,0006468 -logKd/Ki=5.24, IC50=5.8uM IC50=3463nM P41743 16125198 1000 LGLQDFDLLRVIGRGSYAKVLLVRLKKTDRIYAMKVVKKELVNDDEDIDWVQTEKHVFEQASNHPFLVGLHSCFQTESRLFFVIEYVNGGDLMFHMQRQRKLPEEHARFYSAEISLALNYLHERGIIYRDLKLDNVLLDSEGHIKLTDYGMCKEGLRPGDTTSTFCGTPNYIAPEILRGEDYGFSVDWWALGVLMFEMMAGRSPFDQNTEDYLFQVILEKQIRIPRSMSVKAASVLKSFLNKDPKERLGCLPQTGFADIQGHPFFRNVDWDMMEQKQVVPPFKPVQLTPDDDDIVRKIDQSEFEGFEYINPL