1uom A 2.28 BS01 PTI A 1 M343 L346 T347 A350 D351 E353 W383 L387 G521 H524 L525 A546 M37 L40 T41 A44 D45 E47 W77 L81 G215 H218 L219 A231 ? ic50=19nM -logKd/Ki=7.72, IC50=19nM IC50=19nM, EC50=16.5nM P03372 12825935 1547 ALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLESAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKSVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLSSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLPLYDLLLEMLDA