1t4j A 2.7 BS01 FRJ A 1 A189 N193 F196 E200 E276 G277 K279 F280 A189 N193 F196 E200 E276 G277 K279 F280 D181 C215 R221 S222 Q262 D181 C215 R221 S222 Q262 3.1.3.48 0004725,0006470,0016311 -logKd/Ki=5.10, IC50=8uM IC50=8000nM P18031 15258570 299 MEMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIM