1t46 A 1.6 BS01 STI A 1 L595 A621 K623 E640 L644 V668 T670 Y672 C673 I789 H790 R791 L799 C809 D810 F811 L31 A57 K59 E76 L80 V104 T106 Y108 C109 I153 H154 R155 L163 C173 D174 F175 D792 R796 N797 D810 D156 R160 N161 D174 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 -logKd/Ki=6.43, IC50=0.37uM IC50=100nM, Kd=15nM, Ki=14nM, EC50=100nM P10721 15123710 3 GNNYVYIDPTQLPYDHKWEFPRNRLSFGKTLGAGAFGKVVEATAYGLIKSDAAMTVAVKMLKPSAHLTEREALMSELKVLSYLGNHMNIVNLLGACTIGGPTLVITEYCCYGDLLNFLRRKRDSFLALDLEDLLSFSYQVAKGMAFLASKNCIHRDLAARNILLTHGRITKICDFGLARDIKNDSNYVVKGNARLPVKWMAPESIFNCVYTFESDVWSYGIFLWELFSLGSSPYPGMPVDSKFYKMIKEGFRMLSPEHAPAEMYDIMKTCWDADPLKRPTFKQIVQLIEKQISESTN