1o47 A 1.8 BS01 822 A 1 R14 R34 S36 E37 C44 H60 Y61 I73 G95 L96 R14 R34 S36 E37 C44 H60 Y61 I73 G95 L96 2.7.10.2 ic50=4nM -logKd/Ki=8.40, IC50=4nM IC50=5nM P12931 14613321 300 SIQAEEWYFGKITRRESERLLLNAENPRGTFLVRESETTKGAYCLSVSDFDNAKGLNVKHYKIRKLDSGGFYITSRTQFNSLQQLVAYYSKHADGLCHRLTTVCPT