1mx1 A 2.4 BS01 SIA A 1 L1051 G1052 N1079 A1080 T1081 S1082 P1084 Y1118 L31 G32 N59 A60 T61 S62 P64 Y98 G1142 G1143 S1221 A1222 E1354 H1468 G122 G123 S201 A202 E334 H447 3.1.1.1,3.1.1.13,3.1.1.56 0004771,0005737,0005783,0005788,0005811,0005829,0006629,0006695,0008203,0009636,0010875,0010887,0016042,0030855,0042632,0043691,0047374,0051791,0052689,0070857,0071397,0071404,0090122,0090205,0106435,0120188 P23141 12725862 182 SSPPVVDTVHGKVLGKFVSLEGFAQPVAIFLGIPFAKPPLGPLRFTPPQPAEPWSFVKNATSYPPMCTQDPKAGQLLSELFTNRKENIPLKLSEDCLYLNIYTPADLTKKNRLPVMVWIHGGGLMVGAASTYDGLALAAHENVVVVTIQYRLGIWGFFSTGDEHSRGNWGHLDQVAALRWVQDNIASFGGNPGSVTIFGESAGGESVSVLVLSPLAKNLFHRAISESGVALTSVLVKKGDVKPLAEQIAITAGCKTTTSAVMVHCLRQKTEEELLETTLKMKFLSLDLQGDPRESQPLLGTVIDGMLLLKTPEELQAERNFHTVPYMVGINKQEFGWLIPMLMSYPLSEGQLDQKTAMSLLWKSYPLVCIAKELIPEATEKYLGGTDDTVKKKDLFLDLIADVMFGVPSVIVARNHRDAGAPTYMYEFQYRPSFSSDMKPKTVIGDHGDELFSVFGAPFLKEGASEEEIRLSKMVMKFWANFARNGNPNGEGLPHWPEYNQKEGYLQIGANTQAAQKLKDKEVAFWTNLFAK 1mx1 A 2.4 BS02 THA A 1 L1097 F1101 S1221 H1468 L77 F81 S201 H447 G1142 G1143 S1221 A1222 E1354 H1468 G122 G123 S201 A202 E334 H447 3.1.1.1,3.1.1.13,3.1.1.56 0004771,0005737,0005783,0005788,0005811,0005829,0006629,0006695,0008203,0009636,0010875,0010887,0016042,0030855,0042632,0043691,0047374,0051791,0052689,0070857,0071397,0071404,0090122,0090205,0106435,0120188 -logKd/Ki=4.00, Ki>100uM IC50=>100000nM, Ki=>100000nM P23141 12725862 1 SSPPVVDTVHGKVLGKFVSLEGFAQPVAIFLGIPFAKPPLGPLRFTPPQPAEPWSFVKNATSYPPMCTQDPKAGQLLSELFTNRKENIPLKLSEDCLYLNIYTPADLTKKNRLPVMVWIHGGGLMVGAASTYDGLALAAHENVVVVTIQYRLGIWGFFSTGDEHSRGNWGHLDQVAALRWVQDNIASFGGNPGSVTIFGESAGGESVSVLVLSPLAKNLFHRAISESGVALTSVLVKKGDVKPLAEQIAITAGCKTTTSAVMVHCLRQKTEEELLETTLKMKFLSLDLQGDPRESQPLLGTVIDGMLLLKTPEELQAERNFHTVPYMVGINKQEFGWLIPMLMSYPLSEGQLDQKTAMSLLWKSYPLVCIAKELIPEATEKYLGGTDDTVKKKDLFLDLIADVMFGVPSVIVARNHRDAGAPTYMYEFQYRPSFSSDMKPKTVIGDHGDELFSVFGAPFLKEGASEEEIRLSKMVMKFWANFARNGNPNGEGLPHWPEYNQKEGYLQIGANTQAAQKLKDKEVAFWTNLFAK 1mx1 B 2.4 BS01 SIA A 1 K2262 T2278 K241 T257 G2142 G2143 S2221 A2222 E2354 H2468 G121 G122 S200 A201 E333 H446 3.1.1.1,3.1.1.13,3.1.1.56 0004771,0005737,0005783,0005788,0005811,0005829,0006629,0006695,0008203,0009636,0010875,0010887,0016042,0030855,0042632,0043691,0047374,0051791,0052689,0070857,0071397,0071404,0090122,0090205,0106435,0120188 P23141 12725862 182 SPPVVDTVHGKVLGKFVSLEGFAQPVAIFLGIPFAKPPLGPLRFTPPQPAEPWSFVKNATSYPPMCTQDPKAGQLLSELFTNRKENIPLKLSEDCLYLNIYTPADLTKKNRLPVMVWIHGGGLMVGAASTYDGLALAAHENVVVVTIQYRLGIWGFFSTGDEHSRGNWGHLDQVAALRWVQDNIASFGGNPGSVTIFGESAGGESVSVLVLSPLAKNLFHRAISESGVALTSVLVKKGDVKPLAEQIAITAGCKTTTSAVMVHCLRQKTEEELLETTLKMKFLSLDLQGDPRESQPLLGTVIDGMLLLKTPEELQAERNFHTVPYMVGINKQEFGWLIPMLMSYPLSEGQLDQKTAMSLLWKSYPLVCIAKELIPEATEKYLGGTDDTVKKKDLFLDLIADVMFGVPSVIVARNHRDAGAPTYMYEFQYRPSFSSDMKPKTVIGDHGDELFSVFGAPFLKEGASEEEIRLSKMVMKFWANFARNGNPNGEGLPHWPEYNQKEGYLQIGANTQAAQKLKDKEVAFWTNLFAK