1los A 1.9 BS01 UP6 A 1 D20 K42 K72 M126 S127 P180 G202 A203 D18 K40 K70 M124 S125 P178 G196 A197 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=64nM Ki=12400nM O26232 12011084 5001 SRRVDVMDVMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGDPGETLRFADAIIVGASIYLADNPAAAAAGIIESI 1los A 1.9 BS02 UP6 B 1 D75 I76 T79 D73 I74 T77 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=64nM Ki=12400nM O26232 12011084 5002 SRRVDVMDVMNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGDPGETLRFADAIIVGASIYLADNPAAAAAGIIESI 1los B 1.9 BS01 UP6 A 1 D1075 I1076 T1079 D64 I65 T68 K1042 D1070 K1072 D1075 K31 D59 K61 D64 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 Ki=64nM Ki=12400nM O26232 12011084 5001 MNRLILAMDLMNRDDALRVTGEVREYIDTVKIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGDPGETLRFADAIIVGASIYLADNPAAAAAGIIES