1jr1 A 2.6 BS01 IMP A 1 S68 M70 R322 G328 S329 I330 C331 D364 M386 G387 S388 Y411 G413 M414 G415 Q441 G442 S52 M54 R260 G266 S267 I268 C269 D302 M324 G325 S326 Y349 G351 M352 G353 Q363 G364 1.1.1.205 0000166,0003824,0003938,0005634,0005737,0005829,0006164,0006177,0006183,0007623,0016491,0046651,0046872,0071353,0097294 P12269 8681386 1331 GLTAQQLFNCGDGLTYNDFLILPGYIDFTADQVDLTSALTKKITLKTPLVSSPMDTVTEAGMAIAMALTGGIGFIHHNCTPEFQANEVRKVKKYEQGFITDPVVDRVRFEAKMGSRLVIMTKREDLVVAPAGITLKEANEILQRSKLPIVNENDELVAIIARTDLKKNRDYPLASKDAKKQLLCGAAIGTHEDDKYRLDLLALAGVDVVVLDSSQGNSIFQINMIKYMKEKYPNLQVIGGNVVTAAQAKNLIDAGVDALRVGMGCGSICITQEVLACGRPQATAVYKVSEYARRFGVPVIADGGIQNVGHIAKALALGASTVMMGSLLAATTEAPGEYFFSDGIRLKKYRGMGSLDAMIKVAQGVSGAVQDKGSIHKFVPYLIAGIQHSCQDIGAKSLTQVRAMMYSGELKFEKRTSSAQVEGGVHSLHSYEKRLF 1jr1 A 2.6 BS02 MOA A 1 D274 S275 S276 N303 G326 C331 T333 M414 G415 Q441 D212 S213 S214 N241 G264 C269 T271 M352 G353 Q363 1.1.1.205 0000166,0003824,0003938,0005634,0005737,0005829,0006164,0006177,0006183,0007623,0016491,0046651,0046872,0071353,0097294 -logKd/Ki=8.22, Ki=6nM P12269 8681386 1332 GLTAQQLFNCGDGLTYNDFLILPGYIDFTADQVDLTSALTKKITLKTPLVSSPMDTVTEAGMAIAMALTGGIGFIHHNCTPEFQANEVRKVKKYEQGFITDPVVDRVRFEAKMGSRLVIMTKREDLVVAPAGITLKEANEILQRSKLPIVNENDELVAIIARTDLKKNRDYPLASKDAKKQLLCGAAIGTHEDDKYRLDLLALAGVDVVVLDSSQGNSIFQINMIKYMKEKYPNLQVIGGNVVTAAQAKNLIDAGVDALRVGMGCGSICITQEVLACGRPQATAVYKVSEYARRFGVPVIADGGIQNVGHIAKALALGASTVMMGSLLAATTEAPGEYFFSDGIRLKKYRGMGSLDAMIKVAQGVSGAVQDKGSIHKFVPYLIAGIQHSCQDIGAKSLTQVRAMMYSGELKFEKRTSSAQVEGGVHSLHSYEKRLF