Structure of PDB 9cbm Chain R

Receptor sequence
>9cbmR (length=257) Species: 9606,10665 [Search protein sequence]
VTLTLVCLAGLLMLLTVFGNVLVIIAVFTSRALKAPQNLFLVSLASADIL
VATLVIPFSLANEVMGYWYFGKAWCEIYLALDVLFCTSSIVHLCAISLDR
YWSITQAIEYNLKRTPRRIKAIIITVWVISAVISFPEPRCEINDQKWYVI
SSCIGSFFAPCLIMILVYVRIYQIAKRRTRQNREKRFTFVLAVVIGVFVV
CWFPFFFTYTLTAVGCSVPRTLFKFFFWFGYCNSSLNPVIYTIFNHDFRR
AFKKILC
3D structure
PDB9cbm Distinct binding conformations of epinephrine with alpha- and beta-adrenergic receptors.
ChainR
Resolution3.2 Å
3D
structure
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Interaction with ligand
Site
#
Ligand Ligand
chain
Binding residues on receptor
(original residue number in PDB)
Binding residues on receptor
(residue number reindexed from 1)
Binding affinity
BS01 CZX R D128 V129 C132 T133 S215 W402 F405 F406 Y409 F427 D82 V83 C86 T87 S152 W202 F205 F206 Y209 F227
External links
PDB RCSB:9cbm, PDBe:9cbm, PDBj:9cbm
PDBsum9cbm
PubMed39218975
UniProtP00720|ENLYS_BPT4 Endolysin (Gene Name=E);
P08913|ADA2A_HUMAN Alpha-2A adrenergic receptor (Gene Name=ADRA2A)

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