Structure of PDB 4znv Chain B

Receptor sequence
>4znvB (length=243) Species: 9606 (Homo sapiens) [Search protein sequence]
SLALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADREL
VHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLF
APNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILL
NSGVYTFKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLL
ILSHIRHMSNKGMEHLYSMKCKNVVPLSDLLLEMLDAHRLHAP
3D structure
PDB4znv Predictive features of ligand-specific signaling through the estrogen receptor.
ChainB
Resolution1.771 Å
3D
structure
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Enzymatic activity
Enzyme Commision number ?
Interaction with ligand
Site
#
Ligand Ligand
chain
Binding residues on receptor
(original residue number in PDB)
Binding residues on receptor
(residue number reindexed from 1)
Binding affinity
BS01 peptide B I358 K362 Q375 V376 E380 E542 I54 K58 Q71 V72 E76 E233
BS02 4Q7 B E353 L387 M388 L391 F404 G420 M421 I424 H524 L525 E49 L83 M84 L87 F100 G116 M117 I120 H215 L216
External links
PDB RCSB:4znv, PDBe:4znv, PDBj:4znv
PDBsum4znv
PubMed27107013
UniProtP03372|ESR1_HUMAN Estrogen receptor (Gene Name=ESR1)

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