Structure of PDB 2e3k Chain B

Receptor sequence
>2e3kB (length=110) Species: 9606 (Homo sapiens) [Search protein sequence]
HMEQLKHCNGILKELLSKKHAAYAWPFYKPVDASALGLHDYHDIIKHPMD
LSTVKRKMENRDYRDAQEFAADVRLMFSNCYKYNPPDHDVVAMARKLQDV
FEFRYAKMPD
3D structure
PDB2e3k Structural basis for diacetylated histone H4 tail recognition by the second bromodomain of human BRD2
ChainB
Resolution2.3 Å
3D
structure
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Enzymatic activity
Enzyme Commision number ?
Interaction with ligand
Site
#
Ligand Ligand
chain
Binding residues on receptor
(original residue number in PDB)
Binding residues on receptor
(residue number reindexed from 1)
Binding affinity
BS01 peptide B F372 V376 C425 Y428 N429 P430 H433 D434 F27 V31 C80 Y83 N84 P85 H88 D89
External links
PDB RCSB:2e3k, PDBe:2e3k, PDBj:2e3k
PDBsum2e3k
PubMed
UniProtP25440|BRD2_HUMAN Bromodomain-containing protein 2 (Gene Name=BRD2)

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