Structure of PDB 9eyr Chain A

Receptor sequence
>9eyrA (length=239) Species: 7955 (Danio rerio) [Search protein sequence]
HMLSDEQMQIINSLVEAHHKTYDDSYSDFVRFRPPVRRLSMLPHLADLVS
YSIQKVIGFAKMIPGFRDLTAEDQIALLKSSAIEIIMLRSNQSFSLEDMS
WSCGGPDFKYCINDVTKAGHTLELLEPLVKFQVGLKKLKLHEEEHVLLMA
ICLLSPDRPGVQDHVRIEALQDRLCDVLQAYIRIQHPGGRLLYAKMIQKL
ADLRSLNEEHSKQYRSLSFQPEHSMQLTPLVLEVFGSEV
3D structure
PDB9eyr Design, Synthesis, and Biological Evaluation of New Type of Gemini Analogues with a Cyclopropane Moiety in Their Side Chain.
ChainA
Resolution2.56 Å
3D
structure
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Interaction with ligand
Site
#
Ligand Ligand
chain
Binding residues on receptor
(original residue number in PDB)
Binding residues on receptor
(residue number reindexed from 1)
Binding affinity
BS01 peptide A I270 K274 R280 A284 I288 K292 P442 L443 E446 E451 I57 K61 R67 A71 I75 K79 P229 L230 E233 E238
BS02 A1H75 A S265 I299 R302 S303 S306 W314 C316 H333 L337 L341 H423 S52 I86 R89 S90 S93 W101 C103 H120 L124 L128 H210
External links
PDB RCSB:9eyr, PDBe:9eyr, PDBj:9eyr
PDBsum9eyr
PubMed38858308
UniProtQ9PTN2|VDRA_DANRE Vitamin D3 receptor A (Gene Name=vdra)

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