Structure of PDB 9ent Chain A

Receptor sequence
>9entA (length=785) Species: 10116 (Rattus norvegicus) [Search protein sequence]
GSCKGRCFELQEVGPPDCRCDNLCKSYSSCCHDFDELCLKTARGWECTKD
RCGEVRNEENACHCSEDCLSRGDCCTNYQVVCKGESHWVDDDCEEIKVPE
CPAGFVRPPLIIFSVDGFRASYMKKGSKVMPNIEKLRSCGTHAPYMRPVY
PTKTFPNLYTLATGLYPESHGIVGNSMYDPVFDASFHLRGREKFNHRWWG
GQPLWITATKQGVRAGTFFWSVSIPHERRILTILQWLSLPDNERPSVYAF
YSEQPDFSGHKYGPFGPEMTNPLREIDKTVGQLMDGLKQLRLHRCVNVIF
VGDHGMEDVTCDRTEFLSNYLTNVDDITLVPGTLGRIRAKSIKYDPKTII
ANLTCKKPDQHFKPYMKQHLPKRLHYANNRRIEDIHLLVDRRWHVARKPL
DVYKKPSGKCFFQGDHGFDNKVNSMQTVFVGYGPTFKYRTKVPPFENIEL
YNVMCDLLGLKPAPNNGTHGSLNHLLRTNTFRPTMPDEVSRPNYPGIMYL
QSEFDLGCTCDDKKGSTKERHLLYGRPAVLYRTSYDILYHTDFESGYSEI
FLMPLWTSYTISKQAEVSSIPEHLTNCVRPDVRVSPGFSQNCLAYKNDKQ
MSYGFLFPPYLSSSPEAKYDAFLVTNMVPMYPAFKRVWAYFQRVLVKKYA
SERNGVNVISGPIFDYNYDGLRDTEDEIKQYVEGSSIPVPTHYYSIITSC
LDFTQPADKCDGPLSVSSFILPHRPDNDESCNSSEDESKWVEELMKMHTA
RVRDIEHLTGLDFYRKTSRSYSEILTLKTYLHTYE
3D structure
PDB9ent In situ serial crystallography facilitates 96-well plate structural analysis at low symmetry.
ChainA
Resolution2.2 Å
3D
structure
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Interaction with ligand
Site
#
Ligand Ligand
chain
Binding residues on receptor
(original residue number in PDB)
Binding residues on receptor
(residue number reindexed from 1)
Binding affinity
BS01 5JK A L78 Y214 K248 F249 H251 W254 P258 W260 F274 L23 Y159 K193 F194 H196 W199 P203 W205 F219
BS02 ZN A D311 H315 H474 D256 H260 H416
BS03 ZN A D171 T209 D358 H359 D116 T154 D303 H304
BS04 CA A D739 N741 D743 L745 D747 D665 N667 D669 L671 D673
External links
PDB RCSB:9ent, PDBe:9ent, PDBj:9ent
PDBsum9ent
PubMed39008358
UniProtQ64610|ENPP2_RAT Autotaxin (Gene Name=Enpp2)

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