Structure of PDB 8qb0 Chain A

Receptor sequence
>8qb0A (length=113) Species: 9606 (Homo sapiens) [Search protein sequence]
EMQLTPFLILLRKTLEQLQEKDTGNIFSEPVPLSEVPDYLDHIKKPMDFF
TMKQNLEAYRYLNFDDFEEDFNLIVSNCLKYNAKDTIFYRAAVRLREQGG
AVLRQARRQAEKM
3D structure
PDB8qb0 Dual BET/BRPF1 inhibitors induce morphological alteration and cellular death in various human cancer cell lines
ChainA
Resolution1.45 Å
3D
structure
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Interaction with ligand
Site
#		 Ligand Ligand
chain		 Binding residues on receptor
(original residue number in PDB)		 Binding residues on receptor
(residue number reindexed from 1)		 Binding affinity
BS01 Q9U A I652 F653 V657 P658 Y665 Y707 N708 F714 I26 F27 V31 P32 Y39 Y81 N82 F88
External links
PDB RCSB:8qb0, PDBe:8qb0, PDBj:8qb0
PDBsum8qb0
PubMed
UniProtP55201|BRPF1_HUMAN Peregrin (Gene Name=BRPF1)

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