Structure of PDB 5dkg Chain A

Receptor sequence
>5dkgA (length=231) Species: 9606 (Homo sapiens) [Search protein sequence]
NSLALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRE
LVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLL
FAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIIL
LNSGVYTFKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSH
IRHMSNKGMEHLYSMKCPLSDLLLEMLDAHR
3D structure
PDB5dkg Predictive features of ligand-specific signaling through the estrogen receptor.
ChainA
Resolution2.15 Å
3D
structure
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Enzymatic activity
Enzyme Commision number ?
Interaction with ligand
Site
#
Ligand Ligand
chain
Binding residues on receptor
(original residue number in PDB)
Binding residues on receptor
(residue number reindexed from 1)
Binding affinity
BS01 peptide A I358 K362 L372 V376 L379 E380 D538 L539 E542 I55 K59 L69 V73 L76 E77 D221 L222 E225
BS02 5C7 A T347 A350 E353 L387 F404 M421 H524 T44 A47 E50 L84 F101 M118 H211
External links
PDB RCSB:5dkg, PDBe:5dkg, PDBj:5dkg
PDBsum5dkg
PubMed27107013
UniProtP03372|ESR1_HUMAN Estrogen receptor (Gene Name=ESR1)

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