Structure of PDB 4zc9 Chain A

Receptor sequence
>4zc9A (length=127) Species: 9606 (Homo sapiens) [Search protein sequence]
SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVK
LNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNK
PGDDIVLMAEALEKLFLQKINELPTEE
3D structure
PDB4zc9 DRUG DEVELOPMENT. Phthalimide conjugation as a strategy for in vivo target protein degradation.
ChainA
Resolution0.99 Å
3D
structure
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Enzymatic activity
Enzyme Commision number ?
Interaction with ligand
Site
#		 Ligand Ligand
chain		 Binding residues on receptor
(original residue number in PDB)		 Binding residues on receptor
(residue number reindexed from 1)		 Binding affinity
BS01 4MW A W81 P82 L92 L94 N140 I146 M149 W40 P41 L51 L53 N99 I105 M108
External links
PDB RCSB:4zc9, PDBe:4zc9, PDBj:4zc9
PDBsum4zc9
PubMed25999370
UniProtO60885|BRD4_HUMAN Bromodomain-containing protein 4 (Gene Name=BRD4)

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