Structure of PDB 3u5k Chain A

Receptor sequence
>3u5kA (length=126) Species: 9606 (Homo sapiens) [Search protein sequence]
SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVK
LNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNK
PGDDIVLMAEALEKLFLQKINELPTE
3D structure
PDB3u5k Benzodiazepines and benzotriazepines as protein interaction inhibitors targeting bromodomains of the BET family.
ChainA
Resolution1.8 Å
3D
structure
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Enzymatic activity
Enzyme Commision number ?
Interaction with ligand
Site
#		 Ligand Ligand
chain		 Binding residues on receptor
(original residue number in PDB)		 Binding residues on receptor
(residue number reindexed from 1)		 Binding affinity
BS01 08J A W81 P82 V87 L92 I146 W40 P41 V46 L51 I105
External links
PDB RCSB:3u5k, PDBe:3u5k, PDBj:3u5k
PDBsum3u5k
PubMed22137933
UniProtO60885|BRD4_HUMAN Bromodomain-containing protein 4 (Gene Name=BRD4)

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