Structure of PDB 8oeq Chain r Binding Site BS01

Receptor Information
>8oeq Chain r (length=208) Species: 5476 (Candida albicans) [Search protein sequence] [Download receptor structure] [Download structure with residue number starting from 1] [View receptor structure]
ARRPARCYRYCKNKPYPKSRYNRAVPDAKIRIYDLGRKKATVDEFPLCIH
LVSNELEQLSSEALEAARICANKYITKVSGRDSFHLRVRVHPFHVLRINK
MQGMRGAWGKPHGLAARVSIGQIIMSARTKDSNKDVVIEGLRRARYKFPG
QQKIIISKKWGFTPLNRDEYIAKKTNGEVIDDGAYVKFLSRKGNLEANLQ
QFPNYQYS
Ligand information
>8oeq Chain 1 (length=3217) [Search RNA sequence] [Download ligand structure] [Download structure with residue number starting from 1] [View ligand structure]
ugaccucaaaucagguaggacuacccgcugaacuuaagcauaucaauaag
cggaggaaaagaaaccaacagggauugccucaguagcggcgagugaagcg
gcaaaagcucaaauuugaaaucuggcgucuuuggcguccgaguuguaauu
ugaagaagguaucuuugggcccggcucuugucuauguuccuuggaacagg
acgucacagagggugagaaucccgugcgaugagaugacccgggucugugu
aaaguuccuucgacgagucgaguuguuugggaaugcagcucuaagugggu
gguaaauuccaucuaaagcuaaauauuggcgagagaccgauagcgaacaa
guacagugauggaaagaugaaaagaacuuugaaaagagagugaaaaagua
cgugaaauuguugaaagggaagggcuugagaucagacuugguauuuugca
ugcugcgguuuaccgggccagcaucgguuuggagcggcaggauaauggcg
gaggaauguggcacggcuucugcuguguguuauagccucugacgauacug
ccagccuagaccgaggacugcgguuuaccuaggauguuggcauaaugauc
uuaagucgcccgucuugaaacacggaccaaggagucuaacgucuaugcga
guguuuggguguaaaacccguacgcguaaugaaagugaacgaaggugggg
gcccauuagggugcaccaucgaccgauccugauguguucggauggauuug
aguaagagcauagcuguugggacccgaaagauggugaacuaugccugaau
agggugaagccagaggaaacucugguggaggcucguagcgguucugacgu
gcaaaucgaucgucgaauuuggguauaggggcgaaagacuaaucgaacca
ucuaguagcugguuccugccgaaguuucccucaggauagcagaagcucgu
aucaguuuuaugagguaaagcgaaugauuagaagucuugggguugaaaug
accuuaacuuauucucaaacuuuaaauauguaagaaguccuuguugcuua
auugaacguggacaauugaaugaagagcuuuuagugggccauuuuuggua
agcagaacuggcgaugcgggaugaaccgaacgugaaguuaaagugccgga
augcacgcucaucagacaccacaaaagguguuaguucaucuagacagccg
gacgguggccauggaagucggaauccgcuaaggaguguguaacaacucac
cggccgaaugaacuagcccugaaaauggauggcgcucaagcgugcuacuu
auacuucaccgugauugcuguuuugacgcuuucacgaguaggcaggcgug
gaggucagugacgaagccuuugcuguaaagcugggucgaacggccucuag
ugcagaucuuggugguaguagcaaauauucaaaugagaacuuugaagacu
gaaguggggaaagguuccaugucaacagcaguuggacauggguuagucga
uccuaagagauggggaagcuccguuucaacgugcuugauuuuucaggcca
accaucgaaagggaauccgguuaaaauuccggaacuuggauauggauucu
ucacggcaacguaacugaauguggagacgucggcgugagcccugggagga
guuaucuuuucuucuuaacagcuuaucacccuggaauugguuuauccgga
gauggggucuuauggcuggaagagcgcgguaauuuugccgcguccggugc
gcuuacgacgguccuugaaaauccacaggaaggaauaguuuucaugccaa
gucguacucauaaccgcagcaggucuccaagguuaacagccucuaguuga
uagaauaauguagauaagggaagucggcaaaauagauccguaacuucggg
auaaggauuggcucuaaggaucgguuuaacgaucaacuuagaacugguac
ggacaaggggaaucugacugucuaauuaaaacauagcauugugaugguca
gaaagugauguugacacaaugugauuucugcccagugcucugaaugucaa
agugaagaaauucaaccaagcgcggguaaacggcgggaguaacuaugacu
cucuuaagguagccaaaugccucgucaucuaauuagugacgcgcaugaau
ggauuaacgagauucccacugucccuaucuacuaucuagcgaaaccacag
ccaagggaacgggcuuggcagaaucagcggggaaagaagacccuguugag
cuugacucuaguuugacauugugaaaagacauggaggguguagaauaagu
gggagcuucggcgccggugaaauaccacuaccucuauaguuuuuuuacuu
auucaaugaagcggagcuggaggucaaacuccacguucuagcauuaagcc
cucugggcgauccggguugaagacauugucagguggggaguuuggcuggg
gcggcacaucuguuaaacgauaacgcagguguccuaagggggacucaugg
agaacagaaaucuccaguagaacaaaaggguaaaaguccccuugauuuug
auuuucagugugaauacaaaccaugaaaguguggccuaucgauccuuuag
ucccucggaauuugaggcuagaggugccagaaaaguuaccacagggauaa
cuggcuuguggcagucaagcguucauagcgacauugcuuuuugauucuuc
gaugucggcucuuccuaucauaccgaagcagaauucgguaagcguuggau
uguucacccacuaauagggaacgugagcuggguuuagaccgucgugagac
agguuaguuuuacccuacugaugaauguuaucgcaauaguaauugaacuu
aguacgagaggaaccguucauucagauaauugguuuuugcggcugucuga
ucaggcaacgccgcgaagcuaccaucugcuggauuauggcugaacgccuc
uaagucagaauccaugcuagaacgcgaugauuuuugcccugcacauuuua
gauggauacgaauaagacuuuagucgcuggaccauagcaggcuggcaacg
gugcgcuuagcggaaaggcuuugugcgcuugccggcggauagcaauguca
acaugcgcggggauaaauccuuugcauacgacuuagauguacaacggagu
auuguaagcaguagaguagccuuguuguuacgaucugcugagauuaagcu
cuuguugucugauuugu
.......................<<<<<<.....<......>......>>
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(..<<<<<<)))))..]]]....}..........................
...<<....>>...............<<<<....>>>>............
......................<<<<<<<<<<<<.....<<<<.<.<...
......>>.>.>>>..<<<<<<<.<<<<<<<<.<<<<<<<....<<.<<<
<<<<......<<<<<<......>>>>>>.......>>>>>>.>.>>.>>>
>>.>>>>>>>>>>........<<<..>>>.....>>>>>>>....>>>>>
>>>>>>>..<<<<........>>>><<<<<<....<<<<<<.<<<<<<..
<<<..<<<<<.....>>>>>..>>>...<<....>>.......<<<<<..
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.<<<....<<<<<<<....>>>>>>>.....>>>...<<<<.<<.<<...
.....>>>>>>>>....>>>>>>>>>...<<.......>>......>>>>
>>...>..>.>>..<<<<<<....<.<<<....>>>.><<<<<<<<<<..
.<<<.<<<<<<<.....<<<....<<<....<<<<...<<<<<<.....>
>>>>>.>>>>....>>>..>.>>.....>>>>>...<<<<.<<<<.<...
...>>>>>.>>>>.....>>>>>.>>>>>>>>.>>..<<<<.<<<<<...
..>>>>>.>>>>....<<<......>>>...<<<<<<<..<<<<(((...
..<<<<<<.....<<..........<<<.<<<<<<<<<<.......<<<<
<.<<<...<<.........>>...>>>.........<<......>>...>
>>>>...>>>>>>>>>>>>>..........))).>>...>>>>>>.>>>>
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<<<<<<.<<......<<<<..<<<....>>>.>>>>...>>>>>>>>>>.
.>.....>>>>>><<.....<<.....<<<<<<.......>>>>>><<<<
.....<<<<<.<<...<<<<<<...<<.....>>.>>>>>>....((<<<
<<<...<<....<<<....>>>..........<<<<<<....>>>>>>..
....>>....>>>..<<<<<........>>>>>))<<<<.<<<<<<<...
..<<<....>>>.......<<<<<<...<<<<.<<<<<<<.<<<<<<<<<
<..{{{..>>>>>><...<<<<<....<<<<<<....<<<.....>>>..
..>>>>>>.....>>>>>....><<<<<<<......>>>>>>>>>>>...
>>>>>>>.>>>>.........>>>>>>..........>>>..>>>>>>>>
.>>>..>>.....<<......>>>>>>>.<<<<.....>>>>..>>>>..
<<<<.....<<<<<<<.<<.........<.....<<<<<...........
....>>>>><<.<<<<<<<<<<<......>>>>>..>>>>>>.>>.....
.......<<<<<<<<<..<<<.........>>>..<<<<<<<....<<<<
.....>>>>......>>>>>>>...<<..<<<..<<<<<<....<<<...
..<<<<....>>>>.....>>>.>>>>..>>>>><<<<<<.......>>>
>>>........<...........<<<<<.......>>>>>.....>....
.>>....>>.>>>>>>>..>..>>.>>>>>>>..>>>>>>....>>....
<<<<<........>>>>>....[[[[[..{{{.{{......[[[[.{{[[
[[..<<<<<.<<<<<<<<..<<<<<<<<<<...<.<<.............
...............................>>.>...>>>>>>>>>>..
.<<<<<.....<<<<..<<<<<......>>>>>..............<<<
<...>>>>..>>>>..>>>>>.....>>>>>>>>..>>>>>...<<<...
..>>>..<<<<<<...........>>>>>>..<<...<<<<<<<...<<<
<<<.......>>>>>>.....<<...(((>>....>>>>>>>...<<<.<
<<<<.......>>>>.>>>>.<<<....>>>.>>))).......((((((
..((((.>>>>>>))))))))))..........]]]]..}}]]]].....
..<<.<...<<<<<<...<<.......>>...>>>>>>....>.>.>...
....<<<<<.<<<<<<..<.<<<<<<<......>>>>>>>...>.<<<..
.......>>>.....>>>>>..>...>>>.>>....<<<<<<<....>>>
.>>>>....}}..}}}.]]]]]....<<<<<<<<..<<<<...<<<<<..
...............>>>>>..<<<<<...<<<<....<<<<<<<<<<}}
}.>>>>>..>>>>>...>>>>..>>>>>.<<<<...<<<<<.........
..>>>>>...>>>>.>>>>....>>>>>>>>.....<<<<<<.<<<....
...<<..........<<<<..>>>>......>>.......<<<<<<...<
<<<<<<..<<<......>>>..>>>>>>>.>>>>>>..............
..>>>.>>>>>>..<<<<<<<.............>>....<<<<<<<<<.
<<<....<<<<.<..<<<<<......>>>>>..>>>>>...>>>....>>
>>.>>>>>..>>>>>..
Receptor-Ligand Complex Structure
Global viewLocal viewStructure summary

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PDB8oeq Drug-induced rotational movement of the ribosome is a key factor for read-through enhancement
Resolution3.3 Å
Binding residue
(original residue number in PDB)
R3 R4 A6 R7 K13 N14 K15 Y17 Y22 R24 Y34 D35 K39 S61 E63 A64 A67 R88 R90 H92 F94 R98 N100 G114 M115 R116 W119 G120 Q133 R154 Y157 K158 P160 D193 G194 A195 Y196 K198
Binding residue
(residue number reindexed from 1)
R2 R3 A5 R6 K12 N13 K14 Y16 Y21 R23 Y33 D34 K38 S60 E62 A63 A66 R87 R89 H91 F93 R97 N99 G103 M104 R105 W108 G109 Q122 R143 Y146 K147 P149 D182 G183 A184 Y185 K187
External links
PDB RCSB:8oeq, PDBe:8oeq, PDBj:8oeq
PDBsum8oeq
PubMed
UniProtQ5AIB8|RL10_CANAL Large ribosomal subunit protein uL16 (Gene Name=RPL10)

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