Structure of PDB 7to7 Chain E Binding Site BS01

Receptor Information
>7to7 Chain E (length=114) Species: 9606 (Homo sapiens) [Search protein sequence] [Download receptor structure] [Download structure with residue number starting from 1] [View receptor structure]
RKTNQLQYMQNVVVKTLWKHQFAWPFYQPVDAIKLNLPDYHKIIKNPMDM
GTIKKRLENNYYWSASECMQDFNTMFTNCYIYNKPTDDIVLMAQALEKIF
LQKVAQMPQEEVEL
Ligand information
Receptor-Ligand Complex Structure
Global viewLocal viewStructure summary

[Spin on] [Spin off] [Reset]
[High quality] [Low quality]
[White background] [Black background]

[Spin on] [Spin off] [Reset]
[High quality] [Low quality]
[White background] [Black background]
PDB7to7 BRD3-BD1 in complex with RaPID linear peptide 1xAcK.4XE (monoAcK.4xE)
Resolution1.93 Å
Binding residue
(original residue number in PDB)
W57 P58 F59 V63 K67 L68 L70 I122 M125
Binding residue
(residue number reindexed from 1)
W24 P25 F26 V30 K34 L35 L37 I89 M92
Enzymatic activity
Enzyme Commision number ?
External links
PDB RCSB:7to7, PDBe:7to7, PDBj:7to7
PDBsum7to7
PubMed37992806
UniProtQ15059|BRD3_HUMAN Bromodomain-containing protein 3 (Gene Name=BRD3)

[Back to BioLiP]