Structure of PDB 6ulv Chain D Binding Site BS01

Receptor Information
>6ulv Chain D (length=111) Species: 9606 (Homo sapiens) [Search protein sequence] [Download receptor structure] [Download structure with residue number starting from 1] [View receptor structure]
PKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPM
DMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEK
LFLQKINELPT
Ligand information
>6ulv Chain G (length=14) Species: 32630 (synthetic construct) [Search peptide sequence] [Download ligand structure] [Download structure with residue number starting from 1] [View ligand structure]
WKNWCWLKRKLLLR
Receptor-Ligand Complex Structure
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PDB6ulv Cyclic peptides can engage a single binding pocket through highly divergent modes.
Resolution2.2 Å
Binding residue
(original residue number in PDB)
W81 P82 Q85 P86 V87 L92 Y139 I146
Binding residue
(residue number reindexed from 1)
W26 P27 Q30 P31 V32 L37 Y84 I91
Enzymatic activity
Enzyme Commision number ?
External links
PDB RCSB:6ulv, PDBe:6ulv, PDBj:6ulv
PDBsum6ulv
PubMed33046654
UniProtO60885|BRD4_HUMAN Bromodomain-containing protein 4 (Gene Name=BRD4)

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