Structure of PDB 2gpv Chain C Binding Site BS01

Receptor Information
>2gpv Chain C (length=223) Species: 9606 (Homo sapiens) [Search protein sequence] [Download receptor structure] [Download structure with residue number starting from 1] [View receptor structure]
PYNKIVSHLLVAEPEKIYAMPDPTVPDSDIKALTTLCDLADRELVVIIGW
AKHIPGFSTLSLADQMSLLQSAWMEILILGVVYRSLSFEDELVYADDYIM
DEDQSKLAGLLDLNNAILQLVKKYKSMKLEKEEFVTLKAIALANSDSMHI
EDVEAVQKLQDVLHEALQDYEAGQHMEDPRRAGKMLMTLPLLRQTSTKAV
QHFYNIKLEGKVPMHKLFLEMLE
Ligand information
>2gpv Chain I (length=12) Species: 99883 (Tetraodon nigroviridis) [Search peptide sequence] [Download ligand structure] [Download structure with residue number starting from 1] [View ligand structure]
GLEAIIRKALMG
Receptor-Ligand Complex Structure
Global viewLocal viewStructure summary

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PDB2gpv X-ray crystal structures of the estrogen-related receptor-gamma ligand binding domain in three functional states reveal the molecular basis of small molecule regulation.
Resolution2.85 Å
Binding residue
(original residue number in PDB)		I280 K284 M298 W305
Binding residue
(residue number reindexed from 1)		I48 K52 M66 W73
Enzymatic activity
Enzyme Commision number ?
External links
PDB RCSB:2gpv, PDBe:2gpv, PDBj:2gpv
PDBsum2gpv
PubMed16990259
UniProtP62508|ERR3_HUMAN Estrogen-related receptor gamma (Gene Name=ESRRG)

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