Structure of PDB 5u1q Chain B Binding Site BS01

Receptor Information
>5u1q Chain B (length=107) Species: 9606 (Homo sapiens) [Search protein sequence] [Download receptor structure] [Download structure with residue number starting from 1] [View receptor structure]
SAAIHRTQLWFHGRISREESQRLIGQQGLVDGLFLVRESQRNPQGFVLSL
CHLQKVKHYLILPSEEEGRLYFSMDDGQTRFTDLLQLVEFHQLNRGILPC
LLRHCCT
Ligand information
Receptor-Ligand Complex Structure
Global viewLocal viewStructure summary

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PDB5u1q Discovery, Development, and Cellular Delivery of Potent and Selective Bicyclic Peptide Inhibitors of Grb7 Cancer Target.
Resolution2.1 Å
Binding residue
(original residue number in PDB)
R438 K478 H479 Y480 L481 M495
Binding residue
(residue number reindexed from 1)
R17 K57 H58 Y59 L60 M74
Enzymatic activity
Enzyme Commision number ?
External links
PDB RCSB:5u1q, PDBe:5u1q, PDBj:5u1q
PDBsum5u1q
PubMed29083893
UniProtQ14451|GRB7_HUMAN Growth factor receptor-bound protein 7 (Gene Name=GRB7)

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