Structure of PDB 8p9w Chain A Binding Site BS01

Receptor Information
>8p9w Chain A (length=238) Species: 7955 (Danio rerio) [Search protein sequence] [Download receptor structure] [Download structure with residue number starting from 1] [View receptor structure]
HMLSDEQMQIINSLVEAHHKTYDDSYSDFVRFRPPVRLSMLPHLADLVSY
SIQKVIGFAKMIPGFRDLTAEDQIALLKSSAIEIIMLRSNQSFSLEDMSW
SCGGPDFKYCINDVTKAGHTLELLEPLVKFQVGLKKLKLHEEEHVLLMAI
CLLSPDRPGVQDHVRIEALQDRLCDVLQAYIRIQHPGGRLLYAKMIQKLA
DLRSLNEEHSKQYRSLSFQPEHSMQLTPLVLEVFGSEV
Ligand information
Receptor-Ligand Complex Structure
Global viewLocal viewStructure summary

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PDB8p9w A vitamin D-based strategy overcomes chemoresistance in prostate cancer.
Resolution2.9 Å
Binding residue
(original residue number in PDB)
I270 K274 R280 I288 K292 P442 E446 E451
Binding residue
(residue number reindexed from 1)
I56 K60 R66 I74 K78 P228 E232 E237
External links
PDB RCSB:8p9w, PDBe:8p9w, PDBj:8p9w
PDBsum8p9w
PubMed38982588
UniProtQ9PTN2|VDRA_DANRE Vitamin D3 receptor A (Gene Name=vdra)

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