Structure of PDB 7rjp Chain A Binding Site BS01

Receptor Information
>7rjp Chain A (length=127) Species: 9606 (Homo sapiens) [Search protein sequence] [Download receptor structure] [Download structure with residue number starting from 1] [View receptor structure]
SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVK
LNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNK
PGDDIVLMAEALEKLFLQKINELPTEE
Ligand information
Receptor-Ligand Complex Structure
Global viewLocal viewStructure summary

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PDB7rjp Uncovering the Bromodomain Interactome using Site-Specific Azide-Acetyllysine Photochemistry, Proteomic Profiling and Structural Characterization
Resolution1.25 Å
Binding residue
(original residue number in PDB)
W81 V87 L94 Y139 N140 D145 I146
Binding residue
(residue number reindexed from 1)
W40 V46 L53 Y98 N99 D104 I105
Enzymatic activity
Enzyme Commision number ?
External links
PDB RCSB:7rjp, PDBe:7rjp, PDBj:7rjp
PDBsum7rjp
PubMed
UniProtO60885|BRD4_HUMAN Bromodomain-containing protein 4 (Gene Name=BRD4)

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