Structure of PDB 5jhq Chain A Binding Site BS01

Receptor Information
>5jhq Chain A (length=462) Species: 9606 (Homo sapiens) [Search protein sequence] [Download receptor structure] [Download structure with residue number starting from 1] [View receptor structure]
GALRELLEACRNGDVSRVKRLVDAANVNAKDMAGRKSSPLHFAAGFGRKD
VVEHLLQMGANVHARDDGGLIPLHNACSFGHAEVVSLLLCQGADPNARDN
WNYTPLHEAAIKGKIDVCIVLLQHGADPNIRNTDGKSALDLADPSAKAVL
TGEYKKDELLEAARSGNEEKLMALLTPLNVNCHASDGRKSTPLHLAAGYN
RVRIVQLLLQHGADVHAKDKGGLVPLHNACSYGHYEVTELLLKHGACVNA
MDLWQFTPLHEAASKNRVEVCSLLLSHGADPTLVNCHGKSAVDMAPTPEL
RERLTYEFKGHSLLQAAREADLAKVKKTLALEIINFKQPQSHETALHCAV
ASLHPKRKQVTELLLRKGANVNEKNKDFMTPLHVAAERAHNDVMEVLHKH
GAKMNALDTLGQTALHRAALAGHLQTCRLLLSYGSDPSIISLQGFTAAQM
GNEAVQQILSES
Ligand information
Receptor-Ligand Complex Structure
Global viewLocal viewStructure summary

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PDB5jhq Tankyrase-1 Ankyrin Repeats Form an Adaptable Binding Platform for Targets of ADP-Ribose Modification.
Resolution3.2 Å
Binding residue
(original residue number in PDB)
R215 S217 F222 G225 F226 L250 N255 S258 F259 H261 D279 W281 Y283 E288
Binding residue
(residue number reindexed from 1)
R35 S37 F42 G45 F46 L70 N75 S78 F79 H81 D99 W101 Y103 E108
Enzymatic activity
Enzyme Commision number 2.4.2.-
2.4.2.30: NAD(+) ADP-ribosyltransferase.
External links
PDB RCSB:5jhq, PDBe:5jhq, PDBj:5jhq
PDBsum5jhq
PubMed27594684
UniProtO95271|TNKS1_HUMAN Poly [ADP-ribose] polymerase tankyrase-1 (Gene Name=TNKS)

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