Structure of PDB 3v4a Chain A Binding Site BS01
Receptor Information
>3v4a Chain A (length=244) Species:
9606
(Homo sapiens) [
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PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAK
ALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVF
NEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDG
LKNQKFFDELRMNYIKELDRIIACTSCSRRFYQLTKLLDSVQPIARELHQ
FTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTQ
Ligand information
>3v4a Chain B (length=11) Species:
9606
(Homo sapiens) [
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GAFQNLFQSVR
Receptor-Ligand Complex Structure
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PDB
3v4a
Discovery of diarylhydantoins as new selective androgen receptor modulators.
Resolution
1.95 Å
Binding residue
(original residue number in PDB)
V716 K720 Q733 M734 I737 Q738 M894 E897
Binding residue
(residue number reindexed from 1)
V46 K50 Q63 M64 I67 Q68 M219 E222
Enzymatic activity
Enzyme Commision number
?
External links
PDB
RCSB:3v4a
,
PDBe:3v4a
,
PDBj:3v4a
PDBsum
3v4a
PubMed
22897611
UniProt
P10275
|ANDR_HUMAN Androgen receptor (Gene Name=AR)
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