Structure of PDB 3bqd Chain A Binding Site BS01

Receptor Information
>3bqd Chain A (length=253) Species: 9606 (Homo sapiens) [Search protein sequence] [Download receptor structure] [Download structure with residue number starting from 1] [View receptor structure]
LPQLTPTLVSLLEVIEPEVLYAGYDSSVPDSTWRIMTTLNMLGGRQVIAA
VKWAKAIPGFRNLHLDDQMTLLQYSWMSLMAFALGWRSYRQSSANLLCFA
PDLIINEQRMTLPCMYDQCKHMLYVSSELHRLQVSYEEYLCMKTLLLLSS
VPKDGLKSQELFDEIRMTYIKELGKAIVKREGNSSQNWQRFYQLTKLLDS
MHEVVENLLNYCFQTFLDKTMSIEFPEMLAEIITNQIPKYSNGNIKKLLF
HQK
Ligand information
Receptor-Ligand Complex Structure
Global viewLocal viewStructure summary

[Spin on] [Spin off] [Reset]
[High quality] [Low quality]
[White background] [Black background]

[Spin on] [Spin off] [Reset]
[High quality] [Low quality]
[White background] [Black background]
PDB3bqd Doubling the size of the glucocorticoid receptor ligand binding pocket by deacylcortivazol.
Resolution2.5 Å
Binding residue
(original residue number in PDB)
K579 M593 M752 E755
Binding residue
(residue number reindexed from 1)
K55 M69 M228 E231
Enzymatic activity
Enzyme Commision number ?
External links
PDB RCSB:3bqd, PDBe:3bqd, PDBj:3bqd
PDBsum3bqd
PubMed18160712
UniProtP04150|GCR_HUMAN Glucocorticoid receptor (Gene Name=NR3C1)

[Back to BioLiP]