Structure of PDB 2ovh Chain A Binding Site BS01

Receptor Information
>2ovh Chain A (length=243) Species: 9606 (Homo sapiens) [Search protein sequence] [Download receptor structure] [Download structure with residue number starting from 1] [View receptor structure]
IQLIPPLINLLMSIEPDVIYAGHDNTKPDTSSSLLTSLNQLGERQLLSVV
KWSKSLPGFRNLHIDDQITLIQYSWMSLMVFGLGWRSYKHVSGQMLYFAP
DLILNEQRMKESSFYSLCLTMWQIPQEFVKLQVSQEEFLCMKVLLLLNTI
PLEGLRSQTQFEEMRSSYIRELIKAIGLRQKGVVSSSQRFYQLTKLLDNL
HDLVKQLHLYCLNTFIQSRMSEVIAAQLPKILAGMVKPLLFHK
Ligand information
Receptor-Ligand Complex Structure
Global viewLocal viewStructure summary

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PDB2ovh A structural and in vitro characterization of asoprisnil: a selective progesterone receptor modulator.
Resolution2.0 Å
Binding residue
(original residue number in PDB)
V730 K734 R740 I744 I748 I751 Q752 W755
Binding residue
(residue number reindexed from 1)
V50 K54 R60 I64 I68 I71 Q72 W75
Enzymatic activity
Enzyme Commision number ?
External links
PDB RCSB:2ovh, PDBe:2ovh, PDBj:2ovh
PDBsum2ovh
PubMed17356170
UniProtP06401|PRGR_HUMAN Progesterone receptor (Gene Name=PGR)

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