Structure of PDB 1t65 Chain A Binding Site BS01

Receptor Information
>1t65 Chain A (length=251) Species: 9606 (Homo sapiens) [Search protein sequence] [Download receptor structure] [Download structure with residue number starting from 1] [View receptor structure]
CQPIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKW
AKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDL
VFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPV
DGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQP
IARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHT
Q
Ligand information
Receptor-Ligand Complex Structure
Global viewLocal viewStructure summary

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PDB1t65 The Molecular Mechanisms of Coactivator Utilization in Ligand-dependent Transactivation by the Androgen Receptor.
Resolution1.66 Å
Binding residue
(original residue number in PDB)
K717 K720 M734 Q738 E893 E897
Binding residue
(residue number reindexed from 1)
K49 K52 M66 Q70 E225 E229
Enzymatic activity
Enzyme Commision number ?
External links
PDB RCSB:1t65, PDBe:1t65, PDBj:1t65
PDBsum1t65
PubMed15563469
UniProtP10275|ANDR_HUMAN Androgen receptor (Gene Name=AR)

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